Bromide

Bromide

SCHEMBL28137170

Br.O=C(OCCBr)c1ccccc1

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 1/20 0.55
SLC6A3 known ✓ Q01959 1/20 0.55
TDP1 Q9NUW8 2/20 0.68
LMNA P02545 2/20 0.63
MAPK1 P28482 1/20 0.55
HIF1A Q16665 1/20 0.55
KMT2A Q03164 1/20 0.55
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.51
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
TSHR P16473 2/20 0.50
HPGD P15428 1/20 0.50
F2 P00734 1/20 0.50
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
PTPN1 P18031 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL561869 0.98 TDP1 (0.70) TDP1LMNAMAPK1HIF1ASLC6A2
SCHEMBL28488838 0.87 TDP1 (0.54) TDP1LMNAMAPK1SLC6A2SLC6A3
SCHEMBL4111265 0.86 TDP1 (0.85) TDP1LMNAMAPK1HIF1ASLC6A2
SCHEMBL3025063 0.86 TDP1 (0.78) TDP1LMNAMAPK1HIF1ASLC6A2
SCHEMBL137486 0.85 TDP1 (0.83) TDP1LMNAMAPK1HIF1ASLC6A2
SCHEMBL27765449 0.85 TDP1 (0.81) TDP1LMNAMAPK1HIF1ASLC6A2
SCHEMBL14673017 0.85 TDP1 (0.81) TDP1LMNAMAPK1HIF1ASLC6A2
SCHEMBL4230132 0.85 TDP1 (0.81) TDP1LMNAMAPK1HIF1ASLC6A2
SCHEMBL1656434 0.85 TDP1 (0.81) TDP1LMNAMAPK1HIF1ASLC6A2
SCHEMBL547137 0.83 TDP1 (0.79) TDP1LMNAMAPK1HIF1ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104395372-B Conjugated polymer 默克专利股份有限公司 2017-04-05 CN disclosed