SCHEMBL28144690

SCHEMBL28144690

CS(=O)(=O)Cc1nccc(-c2ccccc2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.50
AURKA O14965 1/20 0.50
PRKACA P17612 1/20 0.50
ADORA2A P29274 1/20 0.50
DUSP10 Q9Y6W6 1/20 0.42
IKBKB O14920 1/20 0.42
ASIC3 Q9UHC3 2/20 0.39
MAPT P10636 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
RAB9A P51151 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HSP90AB1 P08238 1/20 0.38
PTK2 Q05397 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
POLB P06746 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10272516 0.78 AURKA (0.53) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL4447801 0.75 BPTF (0.54) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL4101556 0.75 ADORA2A (0.50) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL1514690 0.74 HSP90AA1 (0.58) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL8703546 0.74 AURKA (0.53) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL28145717 0.74 HSP90AA1 (0.53) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL3970473 0.74 AURKA (0.53) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL27293910 0.73 HSP90AA1 (0.49) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL27997667 0.73 HSP90AA1 (0.49) HSP90AA1AURKAPRKACAADORA2ADUSP10
SCHEMBL28144742 0.73 AURKA (0.49) HSP90AA1AURKAPRKACAADORA2ADUSP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106794161-A TrkA kinase inhibitors, composition and its method 默沙东公司 2017-05-31 CN disclosed