SCHEMBL28145308

SCHEMBL28145308

CCc1c(OC(F)(F)F)cccc1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2R P25116 1/20 0.43
MEN1 O00255 1/20 0.42
NR1I2 O75469 1/20 0.42
LMNA P02545 1/20 0.42
CHRM2 P08172 1/20 0.42
CYP3A4 P08684 1/20 0.42
ADRA2A P08913 1/20 0.42
MAPT P10636 1/20 0.42
OPRK1 P41145 1/20 0.42
HTR2B P41595 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KMT2A Q03164 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
KCNK3 O14649 4/20 0.42
KCNK9 Q9NPC2 4/20 0.42
IRAK4 Q9NWZ3 1/20 0.41
SCN9A Q15858 5/20 0.40
HTT P42858 1/20 0.39
PARP1 P09874 1/20 0.39
HCRTR1 O43613 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27574540 0.83 IRAK4 (0.43) F2RMEN1NR1I2LMNACHRM2
SCHEMBL16960407 0.83 F2R (0.40) F2RKCNK3KCNK9HCRTR1HCRTR2
SCHEMBL28152797 0.82 MEN1 (0.43) MEN1NR1I2LMNACHRM2CYP3A4
SCHEMBL1135994 0.81 CTSD (0.49) MEN1NR1I2LMNACHRM2CYP3A4
SCHEMBL18935479 0.80 F2R (0.38) F2RSLC6A3KCNK3KCNK9SCN9A
SCHEMBL16829425 0.80 MEN1 (0.49) MEN1NR1I2LMNACHRM2CYP3A4
SCHEMBL28192692 0.80 KCNK3 (0.45) F2RCYP3A4OPRK1KCNK3KCNK9
SCHEMBL28348750 0.79 MEN1 (0.44) F2RMEN1KMT2AHDAC6KCNK3
SCHEMBL16951289 0.79 F2R (0.38) F2RSLC6A3KCNK3KCNK9HCRTR1
SCHEMBL29710969 0.79 CTNNB1 (0.55) F2RMEN1NR1I2LMNACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106661035-A Pyrazolopyrimidine derivatives as inhibitors of bruton's tyrosine kinase 莱德克斯制药公共有限公司 2017-05-10 CN disclosed