SCHEMBL28147137

SCHEMBL28147137

NC(=O)c1cncnc1.[NaH]

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.56
SIRT2 Q8IXJ6 2/20 0.52
SIRT1 Q96EB6 2/20 0.52
SIRT3 Q9NTG7 2/20 0.52
F7 P08709 1/20 0.52
F3 P13726 1/20 0.52
SARM1 Q6SZW1 1/20 0.52
SIRT6 Q8N6T7 1/20 0.52
SIRT5 Q9NXA8 1/20 0.52
SIRT4 Q9Y6E7 1/20 0.52
AR P10275 1/20 0.43
NNMT P40261 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MKNK1 Q9BUB5 6/20 0.41
MKNK2 Q9HBH9 6/20 0.41
TSHR P16473 2/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
PARP1 P09874 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL503242 0.97
Hydrochloric Acid SCHEMBL25242562 0.95 HCAR2 (0.56) HCAR2SIRT2SIRT1SIRT3F7
Water SCHEMBL27583249 0.95 HCAR2 (0.56) HCAR2SIRT2SIRT1SIRT3F7
SCHEMBL27541990 0.95
Hydrochloric Acid SCHEMBL12971394 0.95 HCAR2 (0.56) HCAR2SIRT2SIRT1SIRT3F7
SCHEMBL27941587 0.95 HCAR2 (0.56) HCAR2SIRT2SIRT1SIRT3F7
Hydrochloric Acid SCHEMBL28749975 0.92 HCAR2 (0.54) HCAR2SIRT2SIRT1SIRT3F7
Sulfuric Acid SCHEMBL27952916 0.88 HCAR2 (0.50) HCAR2SIRT2SIRT1SIRT3F7
Formic Acid SCHEMBL25244373 0.88 HCAR2 (0.50) HCAR2SIRT2SIRT1SIRT3F7
SCHEMBL27941661 0.84 HCAR2 (0.46) HCAR2SIRT2SIRT1SIRT3F7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109923117-A Use the combination therapy of the phosphoinositide 3-kinase inhibitor with zinc bound fraction 柯瑞斯公司 2019-06-21 CN disclosed
CN-105461736-B Inhibitors of phosphatidylinositol3 3-kinase with zinc bound site 柯瑞斯公司 2018-06-12 CN disclosed
CN-104292242-B Pyrantel compound and preparation, as well as preparation method and application of pyrantel compound and preparation 广州必贝特医药技术有限公司 2017-05-17 CN disclosed
CN-105461736-A PHOSPHOINOSITIDE 3-KINASE INHIBITOR WITH A ZINC BINDING MOIETY CURIS INC 2016-04-06 CN disclosed
CN-103582483-B Phosphatidylinositol 3-kinase inhibitors with zinc binding sites CURIS, INC. (US) 2016-02-17 CN disclosed
CN-103582483-A Phosphatidylinositol 3-kinase inhibitors with zinc binding sites CURIS INC 2014-02-12 CN disclosed