SCHEMBL28147642

SCHEMBL28147642

COc1ccc(CNC(=O)C(N)Cc2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.60
RAB9A P51151 2/20 0.56
ALDH1A1 P00352 2/20 0.55
CTSD P07339 2/20 0.54
CARM1 Q86X55 1/20 0.54
PRMT6 Q96LA8 1/20 0.54
KMT2A Q03164 1/20 0.54
TSHR P16473 2/20 0.53
CASR P41180 1/20 0.53
PLA2G1B P04054 1/20 0.52
ATG4B Q9Y4P1 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16254370 1.00 NPC1 (0.60) NPC1RAB9AALDH1A1CTSDCARM1
SCHEMBL15892590 1.00 NPC1 (0.60) NPC1RAB9AALDH1A1CTSDCARM1
Hydrochloric Acid SCHEMBL15881247 0.99 NPC1 (0.59) NPC1RAB9AALDH1A1CTSDCARM1
Hydrochloric Acid SCHEMBL17335540 0.99 NPC1 (0.59) NPC1RAB9AALDH1A1CTSDCARM1
Hydrochloric Acid SCHEMBL20473203 0.99 NPC1 (0.59) NPC1RAB9AALDH1A1CTSDCARM1
SCHEMBL18492928 0.88 GAA (0.59) ALDH1A1CARM1PRMT6KMT2A
SCHEMBL7413310 0.87 ALPI (0.61) ALDH1A1KMT2A
SCHEMBL3114367 0.87 ALPI (0.61) ALDH1A1KMT2A
SCHEMBL13073347 0.87 KMT2A (0.63) NPC1RAB9AALDH1A1KMT2A
SCHEMBL21582601 0.87 ALDH1A1 (0.60) NPC1RAB9AALDH1A1CARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108368133-A Urea peptidomimetic boronic acid compounds and its pharmaceutical composition, preparation method and purposes 北京大学 2018-08-03 CN disclosed
CN-106588965-A Urea peptidomimetic boric acid compound as well as pharmaceutical composition, preparation method and application thereof 北京大学 2017-04-26 CN disclosed