SCHEMBL28148792

SCHEMBL28148792

O=S(=O)(c1ccccc1)c1ccc(CN2CC=Cc3ccccc32)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.41
NAMPT P43490 1/20 0.40
TYMS P04818 3/20 0.39
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
SRC P12931 3/20 0.38
PRKACA P17612 1/20 0.38
PRKACG P22612 1/20 0.38
PRKACB P22694 1/20 0.38
KDM4E B2RXH2 2/20 0.37
MAPT P10636 2/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30167783 0.85 NAMPT (0.44) NAMPTTYMSCYP3A4CYP2D6CYP2C9
SCHEMBL28148757 0.85 NAMPT (0.44) NAMPTTYMSCYP3A4CYP2D6CYP2C9
SCHEMBL27540773 0.84 EPHX2 (0.41) CYP2D6CYP2C9CYP2C19L3MBTL1KMT2A
Hydrochloric Acid SCHEMBL28844174 0.82 EPHX2 (0.40) CYP2D6CYP2C9CYP2C19L3MBTL1KMT2A
Bromide SCHEMBL28875349 0.82 EPHX2 (0.40) CYP2D6CYP2C9CYP2C19L3MBTL1KMT2A
SCHEMBL28844956 0.81 NAMPT (0.40) HTR6NAMPTTYMSPSEN1PSEN2
SCHEMBL30167580 0.81 NAMPT (0.40) HTR6NAMPTTYMSPSEN1PSEN2
SCHEMBL28641047 0.79 EPHX2 (0.37) CYP2D6CYP2C9CYP2C19L3MBTL1KMT2A
SCHEMBL28149958 0.77 TYMS (0.41) HTR6NAMPTTYMSSRCPRKACA
SCHEMBL27542961 0.77 EPHX2 (0.36) CYP2D6CYP2C9CYP2C19L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103384668-B compounds and compositions for inhibition of NAMPT 福马TM有限责任公司 2017-05-31 CN claimed