SCHEMBL28148757

SCHEMBL28148757

O=S(=O)(c1ccccc1)c1ccc(CN2CC=Cc3cnccc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 15/20 0.44
CYP2C9 P11712 3/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 1/20 0.44
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
TYMS P04818 3/20 0.38
USP2 O75604 1/20 0.37
TP53 P04637 1/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30167783 1.00 NAMPT (0.44) NAMPTCYP2C9CYP2D6CYP2C19CA12
SCHEMBL28148792 0.85 HTR6 (0.41) NAMPTCYP2C9CYP2D6CYP2C19TYMS
SCHEMBL28148791 0.84 NAMPT (0.46) NAMPTUSP2TSHR
SCHEMBL30167576 0.84 NAMPT (0.46) NAMPTUSP2TSHR
SCHEMBL30167580 0.78 NAMPT (0.40) NAMPTTYMSUSP2TSHR
SCHEMBL28844956 0.78 NAMPT (0.40) NAMPTTYMSUSP2TSHR
SCHEMBL30167572 0.75 NAMPT (0.43) NAMPTCYP2C9CYP2D6CYP2C19CA12
SCHEMBL28203325 0.73 CACNA1I (0.34) CYP2C9CYP2D6USP2TP53CYP3A4
SCHEMBL28149958 0.69 TYMS (0.41) NAMPTCYP2C9CYP2D6CYP2C19TYMS
SCHEMBL27540773 0.69 EPHX2 (0.41) CYP2C9CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103384668-B compounds and compositions for inhibition of NAMPT 福马TM有限责任公司 2017-05-31 CN claimed