SCHEMBL28153265

SCHEMBL28153265

Cc1cccc(C)c1NC(=O)C1CCCCC1=O

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.52
CYP1A2 P05177 1/20 0.51
RECQL P46063 1/20 0.51
KCNK3 O14649 1/20 0.50
LMNA P02545 1/20 0.50
MCL1 Q07820 1/20 0.50
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
KCNH2 Q12809 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
ALOX12 P18054 1/20 0.46
SCN1A P35498 1/20 0.45
SCN2A Q99250 1/20 0.45
SCN3A Q9NY46 1/20 0.45
MAPK1 P28482 1/20 0.44
POLB P06746 1/20 0.44
ALDH1A1 P00352 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22430578 0.76 MEN1 (0.64) EPHX1KCNK3LMNACYP3A4CYP2D6
SCHEMBL8008669 0.75 GRK2 (0.61) CYP1A2RECQLMCL1KMT2AALDH1A1
SCHEMBL22423670 0.75 MEN1 (0.68) EPHX1KCNK3LMNAMEN1KMT2A
SCHEMBL23835701 0.75 EPHX1 (0.55) EPHX1KCNK3LMNACYP3A4CYP2D6
SCHEMBL10742560 0.74 CYP1A2 (0.68) EPHX1CYP1A2RECQLLMNAMCL1
SCHEMBL1719455 0.74 MCL1 (0.64) CYP1A2MCL1MEN1KMT2AMAPK1
SCHEMBL12821059 0.72 MCL1 (0.54) CYP1A2RECQLMCL1MEN1KMT2A
SCHEMBL14826669 0.72 MEN1 (0.52) EPHX1KCNK3LMNACYP3A4CYP2D6
SCHEMBL2616379 0.72 EPHX1 (0.51) EPHX1KCNK3LMNACYP3A4CYP2D6
SCHEMBL3261012 0.72 EPHX1 (0.51) EPHX1KCNK3LMNACYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106928126-B Amide derivative, preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2019-12-20 CN disclosed
CN-106928126-A A kind of amide derivatives and preparation method thereof and application pharmaceutically 四川海思科制药有限公司 2017-07-07 CN disclosed