SCHEMBL28154232

SCHEMBL28154232

Brc1ccc(-c2ncnc(-c3cccs3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 12/20 0.49
RAB9A P51151 12/20 0.49
SMN1; SMN2 Q16637 9/20 0.49
MAPT P10636 7/20 0.49
KDM4E B2RXH2 7/20 0.49
ALDH1A1 P00352 5/20 0.49
HPGD P15428 4/20 0.49
TDP1 Q9NUW8 3/20 0.49
HSD17B10 Q99714 2/20 0.49
TSHR P16473 1/20 0.49
CASP3 P42574 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
ATM Q13315 2/20 0.47
PKM P14618 1/20 0.43
ABL1 P00519 1/20 0.43
BCR P11274 1/20 0.43
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28772850 0.85 NPC1 (0.46) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL27110794 0.84 KDM4E (0.50) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL28154237 0.83 RAB9A (0.44) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL28135933 0.79 SMN1; SMN2 (0.73) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL13930812 0.77 NPC1 (0.75) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL474978 0.77 NPC1 (0.60) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL28451522 0.75 NPC1 (0.63) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL28409729 0.75 NPC1 (0.63) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL1310724 0.74 ABL1 (0.60) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL28467605 0.74 RAB9A (0.47) NPC1RAB9ASMN1; SMN2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106866563-B Method for preparing 2, 4-disubstituted-1, 3,5 triazine derivative 中国科学院大连化学物理研究所 2020-02-14 CN disclosed
CN-106866563-A A kind of method for preparing the pyrrolotriazine derivatives of bis- substitutions of 2,4- -1,3,5 中国科学院大连化学物理研究所 2017-06-20 CN disclosed