SCHEMBL28155449

SCHEMBL28155449

OCCc1ccc(CN2CCN(c3ccccc3)CC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 5/20 0.72
DRD2 P14416 3/20 0.58
HTR1A P08908 1/20 0.58
DRD3 P35462 2/20 0.57
SIGMAR1 Q99720 3/20 0.55
HTR7 P34969 1/20 0.55
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
HTT P42858 1/20 0.54
ADRA1D P25100 1/20 0.53
ADRA1A P35348 1/20 0.53
ADRA1B P35368 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3242189 0.87 DRD4 (0.77) DRD4DRD2HTR1ADRD3SIGMAR1
SCHEMBL6031812 0.84 DRD4 (1.00) DRD4DRD2HTR1ADRD3SIGMAR1
SCHEMBL6221968 0.84 DRD4 (0.72) DRD4DRD2HTR1ADRD3SIGMAR1
SCHEMBL9720693 0.83 DRD4 (0.87) DRD4DRD2DRD3SIGMAR1HTR7
SCHEMBL3320211 0.82 DRD4 (0.74) DRD4DRD2DRD3SIGMAR1HTR7
SCHEMBL12861757 0.81 DRD4 (0.79) DRD4DRD2HTR1ADRD3SIGMAR1
SCHEMBL4649494 0.81 DRD4 (0.87) DRD4DRD2DRD3SIGMAR1KDM4E
SCHEMBL22532699 0.81 DRD4 (0.79) DRD4DRD2HTR1ADRD3SIGMAR1
SCHEMBL10713886 0.80 DRD4 (0.66) DRD4DRD2DRD3SIGMAR1HTR7
SCHEMBL13959204 0.80 HTR1A (0.71) DRD4DRD2HTR1ASIGMAR1ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106957280-B Ether-type aryl bridged piperazine derivatives and its salt, preparation method and the purposes in preparation treatment anti-tumor drug 洛阳师范学院 2019-02-15 CN disclosed
CN-106957280-A Ether-type aryl bridged piperazine derivatives and its salt, preparation method and the purposes in treatment antineoplastic is prepared 洛阳师范学院 2017-07-18 CN disclosed