SCHEMBL28162172

SCHEMBL28162172

N#Cc1cccc(=O)n1F

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
MEN1 O00255 1/20 0.31
PKM P14618 1/20 0.31
KMT2A Q03164 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
ALOX15 P16050 1/20 0.30
MAPK1 P28482 1/20 0.30
MCL1 Q07820 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17610033 0.74 MEN1 (0.41) MEN1PKMKMT2A
SCHEMBL27876356 0.74 MEN1 (0.31) MEN1PKMKMT2ACA1CA2
SCHEMBL26750150 0.66 GRM2 (0.38) GRIN1GRIN2AMEN1PKMKMT2A
SCHEMBL27977646 0.65
SCHEMBL7235617 0.58 AR (0.32) MAPTHPGDALOX15MCL1HSD17B10
SCHEMBL7072277 0.58 GLA (0.37) KDM4EALDH1A1MAPTHPGDALOX15
SCHEMBL7233666 0.56
SCHEMBL27431673 0.56 LMNA (0.36) ALDH1A1MAPT
SCHEMBL25596832 0.56
SCHEMBL3934072 0.56

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107001328-A Pyridin-2 (1H) -one quinolinone derivatives as mutant isocitrate dehydrogenase inhibitors 福马治疗股份有限公司 2017-08-01 CN disclosed