SCHEMBL28166240

SCHEMBL28166240

Oc1cccc(CN2CCOCC2)c1Cl

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 8/20 0.71
CYP2C9 P11712 2/20 0.57
ALOX15 P16050 1/20 0.57
HSD17B10 Q99714 1/20 0.57
MPO P05164 1/20 0.51
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
KDM4E B2RXH2 3/20 0.49
KMT2A Q03164 3/20 0.49
ALDH1A1 P00352 3/20 0.49
MAPT P10636 2/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
POLB P06746 1/20 0.49
MEN1 O00255 1/20 0.49
CXCR4 P61073 1/20 0.47
METAP2 P50579 1/20 0.47
NPC1 O15118 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28662303 0.85 CYP2A13 (0.59) CYP2A13CYP2C9ALOX15HSD17B10MPO
SCHEMBL3378848 0.85 KDM4E (0.67) CYP2A13MPOCYP2D6CYP2C19KDM4E
SCHEMBL10665335 0.83 KDM4E (0.70) CYP2A13MPOCYP2D6CYP2C19KDM4E
SCHEMBL4105461 0.83 CYP2A13 (1.00) CYP2A13CYP2C9ALOX15HSD17B10KDM4E
SCHEMBL4327006 0.83 MPO (0.75) CYP2A13CYP2C9ALOX15HSD17B10MPO
SCHEMBL10787841 0.81 MPO (0.72) CYP2A13CYP2C9ALOX15HSD17B10MPO
SCHEMBL7114819 0.81 KDM4E (0.64) CYP2A13CYP2C9ALOX15HSD17B10CYP3A4
SCHEMBL13849993 0.81 CYP2A13 (0.71) CYP2A13CYP2C9ALOX15HSD17B10KDM4E
SCHEMBL18190587 0.81 CYP2A13 (0.71) CYP2A13CYP2C9ALOX15HSD17B10CYP3A4
SCHEMBL18190447 0.81 CYP2A13 (0.71) CYP2A13CYP2C9ALOX15HSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107082782-A Substituted xanthine and its application method 海德拉生物科学有限公司 2017-08-22 CN disclosed
CN-105143229-B Substituted xanthines and methods of use thereof 海德拉生物科学有限公司 2017-06-30 CN disclosed