SCHEMBL28177002

SCHEMBL28177002

CC1Cc2ccccc2C(Cl)=N1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 9/20 0.62
NOS2 P35228 7/20 0.62
ACHE P22303 1/20 0.44
TSHR P16473 1/20 0.41
METAP1 P53582 1/20 0.34
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10481212 0.78 NOS3 (0.65) NOS3NOS2ACHETSHRMETAP1
SCHEMBL8060964 0.77 NOS3 (1.00) NOS3NOS2ACHETSHR
SCHEMBL11742766 0.77 NOS3 (0.62) NOS3NOS2ACHETSHRMETAP1
Iodide SCHEMBL8098294 0.76 NOS3 (0.96) NOS3NOS2ACHETSHR
Hydrochloric Acid SCHEMBL9530199 0.75 NOS3 (0.56) NOS3NOS2ACHETSHRMETAP1
SCHEMBL5418672 0.73 TSHR (0.49) NOS3NOS2ACHETSHRHTR2A
SCHEMBL11750271 0.73 NOS3 (0.62) NOS3NOS2ACHETSHRMETAP1
SCHEMBL18644310 0.72 NOS3 (0.56) NOS3NOS2ACHETSHRHTR1A
SCHEMBL11745091 0.72 NOS3 (0.56) NOS3NOS2ACHETSHRMETAP1
SCHEMBL8099687 0.70 NOS3 (0.54) NOS3NOS2ACHETSHRMETAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107207464-B Substituted dihydro-isoquinoline ketone compound 辉瑞大药厂 2019-10-22 CN disclosed
CN-107207464-A Substituted dihydro-isoquinoline assimilation compound 辉瑞大药厂 2017-09-26 CN disclosed