SCHEMBL28178783

SCHEMBL28178783

Fc1ccc(-c2ccc3ncncc3c2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.61
PIK3CD O00329 1/20 0.61
EGFR P00533 6/20 0.53
MAP4K4 O95819 3/20 0.50
FGFR4 P22455 1/20 0.49
TDO2 P48775 1/20 0.48
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
CDK8 P49336 1/20 0.42
CLK2 P49760 1/20 0.42
CDK7 P50613 1/20 0.42
CDK9 P50750 1/20 0.42
CDK5 Q00535 1/20 0.42
ACVR1 Q04771 1/20 0.42
ROCK1 Q13464 1/20 0.42
DYRK1A Q13627 1/20 0.42
LRRK2 Q5S007 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
CYP1A2 P05177 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8644295 0.89 PIK3CA (0.73) PIK3CAPIK3CDEGFRMAP4K4FGFR4
SCHEMBL17410801 0.85 EGFR (0.60) PIK3CAPIK3CDEGFRFGFR4TDO2
SCHEMBL29891394 0.85 EGFR (0.60) PIK3CAPIK3CDEGFRFGFR4TDO2
SCHEMBL28298099 0.85 PIK3CA (0.65) PIK3CAPIK3CDEGFRMAP4K4FGFR4
SCHEMBL3042419 0.84 PIK3CD (0.63) PIK3CAPIK3CDEGFRMAP4K4FGFR4
SCHEMBL20687402 0.84 PIK3CD (0.73) PIK3CAPIK3CDEGFRMAP4K4FGFR4
SCHEMBL3535171 0.82 PIK3CA (0.61) PIK3CAPIK3CDEGFRMAP4K4FGFR4
SCHEMBL28292972 0.82 PIK3CA (0.61) PIK3CAPIK3CDEGFRMAP4K4FGFR4
SCHEMBL28158032 0.78 EGFR (0.76) PIK3CAPIK3CDEGFRMAP4K4FGFR4
SCHEMBL27597718 0.78 PIK3CA (0.56) PIK3CAPIK3CDEGFRMAP4K4FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104507933-B Amido quinazoline and Pyridopyrimidine derivatives 霍夫曼-拉罗奇有限公司 2017-10-31 CN disclosed