SCHEMBL28298099

SCHEMBL28298099

Fc1cccc(-c2ccc3ncncc3c2)c1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.65
PIK3CD O00329 1/20 0.65
MAP4K4 O95819 4/20 0.54
EGFR P00533 5/20 0.49
TDO2 P48775 1/20 0.48
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 3/20 0.47
USP2 O75604 2/20 0.47
TSHR P16473 2/20 0.47
ALDH1A1 P00352 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
FGFR4 P22455 1/20 0.46
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD17B10 Q99714 1/20 0.44
NT5E P21589 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30568954 0.91 PIK3CA (0.58) PIK3CAPIK3CDMAP4K4EGFRTDO2
SCHEMBL28178783 0.85 PIK3CA (0.61) PIK3CAPIK3CDMAP4K4EGFRTDO2
SCHEMBL8644295 0.84 PIK3CA (0.73) PIK3CAPIK3CDMAP4K4EGFRTDO2
SCHEMBL28139430 0.84 PIK3CA (0.48) PIK3CAPIK3CDMAP4K4TDO2CYP1A2
SCHEMBL20687402 0.83 PIK3CD (0.73) PIK3CAPIK3CDMAP4K4EGFRTDO2
SCHEMBL17410801 0.81 EGFR (0.60) PIK3CAPIK3CDEGFRTDO2FGFR4
SCHEMBL29891394 0.81 EGFR (0.60) PIK3CAPIK3CDEGFRTDO2FGFR4
SCHEMBL28178788 0.81 EGFR (0.67) PIK3CAPIK3CDMAP4K4EGFRTDO2
SCHEMBL28156873 0.81 PDGFRB (0.55) PIK3CAPIK3CDMAP4K4EGFRPDGFRB
SCHEMBL30568937 0.79 TDO2 (0.53) PIK3CAPIK3CDMAP4K4EGFRTDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843858-A Certain chemical entities, composition and method 润新生物公司 2019-06-04 CN disclosed