SCHEMBL28182902

SCHEMBL28182902

O=C(Nc1ccc(Cl)c(C(F)(F)F)c1)Nc1c(F)cc(O)cc1F

nearest known ligand 0.74

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.74
TRPV1 Q8NER1 12/20 0.69
CA1 P00915 4/20 0.58
CA2 P00918 4/20 0.58
CA7 P43166 4/20 0.58
CA9 Q16790 4/20 0.58
PDK1 Q15118 1/20 0.56
HDAC1 Q13547 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12320168 0.87 KDR (0.70) KDRTRPV1CA1CA2CA7
SCHEMBL29364392 0.86 KDR (1.00) KDRTRPV1CA1CA2CA7
SCHEMBL118026 0.86 KDR (1.00) KDRTRPV1CA1CA2CA7
SCHEMBL281864 0.85 KDR (0.85) KDRTRPV1CA1CA2CA7
SCHEMBL21751016 0.84 KDR (0.78) KDRTRPV1CA1CA2CA7
SCHEMBL22092657 0.83 KDR (0.82) KDRTRPV1CA1CA2CA7
SCHEMBL29494948 0.83 KDR (0.82) KDRTRPV1CA1CA2CA7
SCHEMBL16884950 0.82 KDR (0.85) KDRTRPV1CA1CA2CA7
SCHEMBL9084296 0.82 KDR (0.85) KDRTRPV1CA1CA2CA7
SCHEMBL4548158 0.82 KDR (0.90) KDRTRPV1CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111718294-A Crystal form of medicine for treating intestinal cancer 北京康立生医药技术开发有限公司 2020-09-29 CN claimed
CN-111718294-A Crystal form of medicine for treating intestinal cancer 北京康立生医药技术开发有限公司 2020-09-29 CN disclosed
CN-107382845-A A kind of compound for treating intestinal cancer 姜才华 2017-11-24 CN disclosed
CN-107375282-A A kind of pharmaceutical preparation for treating intestinal cancer 姜才华 2017-11-24 CN disclosed
CN-107362163-A A kind of pharmaceutical preparation for treating intestinal cancer 黄才华 2017-11-21 CN disclosed