SCHEMBL28185286

SCHEMBL28185286

O=C(Cl)c1ccc(-c2cnccn2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
PIM2 Q9P1W9 2/20 0.46
PIM1 P11309 1/20 0.46
NPY5R Q15761 1/20 0.45
KMO O15229 1/20 0.42
DHODH Q02127 1/20 0.42
ABL1 P00519 1/20 0.41
P2RX7 Q99572 3/20 0.41
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
POLB P06746 1/20 0.40
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PI4KA P42356 1/20 0.40
PIK3CG P48736 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31227217 0.84 PIM2 (0.45) PIM2PIM1ABL1HDAC3HDAC1
SCHEMBL16995118 0.79 PIM2 (0.52) PIM2PIM1NPY5RKMODHODH
SCHEMBL6960490 0.79 NPY5R (0.65) PIM2PIM1NPY5RKMOPIK3CD
SCHEMBL16291541 0.76 CYP2D6 (0.45) MKNK1MKNK2PIM2PIM1DHODH
SCHEMBL25326508 0.74 KMO (0.49) NPY5RKMOP2RX7PIK3CDPIK3CA
SCHEMBL12492145 0.74 CYP3A4 (0.52) PIM2PIM1NPY5RKMOHDAC3
SCHEMBL23535785 0.73 PIM2 (0.56) PIM2PIM1KMODHODHABL1
SCHEMBL1027774 0.73 GAA (0.45) MKNK1MKNK2
Hydrochloric Acid SCHEMBL2841145 0.71 GAA (0.43) MKNK1MKNK2
SCHEMBL28925103 0.71 MKNK1 (0.49) MKNK1MKNK2PIM2PIM1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107427699-A For treating the KDM1A inhibitor of disease 伊美格生物科学公司 2017-12-01 CN disclosed