SCHEMBL28186243

SCHEMBL28186243

O=[N+]([O-])c1conc1-c1ccccc1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EIF4E P06730 1/20 0.38
NOTUM Q6P988 2/20 0.38
PSMB8 P28062 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
MYC P01106 1/20 0.36
MAX P61244 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HSD11B1 P28845 1/20 0.36
CRHR1 P34998 1/20 0.35
C1R P00736 1/20 0.35
SCN9A Q15858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ABCC8 Q09428 2/20 0.34
KCNJ11 Q14654 2/20 0.34
MASP2 O00187 1/20 0.34
F2 P00734 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28185540 0.81 NPC1 (0.40) EIF4ECYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL28853237 0.78 ALDH1A1 (0.40) CYP1A2CYP3A4CYP2C19ALDH1A1MYC
SCHEMBL6371400 0.75 ALDH1A1 (0.53) EIF4ECYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL28186239 0.74 ALDH1A1 (0.53) ALDH1A1POLBTDP1L3MBTL1
SCHEMBL15428680 0.74 DPP4 (0.42) NOTUMPSMB8HSD11B1C1RSCN9A
SCHEMBL28186260 0.74 MAPT (0.45) CYP3A4ALDH1A1POLBMYCMAX
SCHEMBL28186241 0.74 NOTUM (0.39) NOTUMPSMB8ALDH1A1HSD11B1C1R
SCHEMBL7918730 0.73 ABCC1 (0.49) ALDH1A1MYCTDP1ABCC8KCNJ11
SCHEMBL27860631 0.72 ALDH1A1 (0.46) NOTUMPSMB8ALDH1A1POLBC1R
SCHEMBL28185546 0.72 SCN2A (0.44) EIF4ENOTUMCYP3A4ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107382892-A A kind of preparation technology of the nitro isoxazole compound of 3 aryl 4 贵州大学 2017-11-24 CN disclosed