SCHEMBL28190043

SCHEMBL28190043

CC(C)(C)OC(=O)Nc1cc(C(=O)O)c(Br)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
LCK P06239 1/20 0.40
FYN P06241 1/20 0.40
ATR Q13535 1/20 0.38
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27214502 0.83 CA12 (0.42) CA12CA1CA2CA9ATR
SCHEMBL22987101 0.82 HPGD (0.50) HSD17B10MEN1NPC1HTTRAB9A
SCHEMBL29840249 0.82 AAK1 (0.46) CA12CA1CA2CA9ATR
SCHEMBL22987099 0.79 HTT (0.41) CA12CA1CA2CA9ATR
SCHEMBL6250449 0.79 SMN1; SMN2 (0.43) ATRTSHRHSD17B10MEN1NPC1
SCHEMBL13247607 0.79 CA12 (0.43) CA12CA1CA2CA9LCK
SCHEMBL31497650 0.77 ATR (0.54) CA12CA1CA2CA9ATR
SCHEMBL20158012 0.77 PPARG (0.40) NPC1RAB9AKMT2AHSP90AA1HSP90AB1
SCHEMBL20157982 0.76 LCK (0.39) LCKNPC1HTTRAB9ARXFP1
SCHEMBL458679 0.75 AAK1 (0.46) ATRNPC1RAB9AHSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104470925-B Imidazo-triazine formonitrile HCN as kinase inhibitor 百时美施贵宝公司 2017-12-05 CN disclosed