SCHEMBL281926

SCHEMBL281926

O=C(Nc1ccc(Oc2ncnc3cc(F)ccc23)cc1)NN(C(=O)Nc1ccc(Oc2ncnc3cc(F)ccc23)cc1)c1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 15/20 0.58
RAF1 P04049 4/20 0.54
KDR P35968 3/20 0.54
PDGFRB P09619 2/20 0.54
KIT P10721 2/20 0.54
PDGFRA P16234 2/20 0.54
FLT3 P36888 2/20 0.54
FGFR2 P21802 1/20 0.54
BRAF P15056 4/20 0.53
AURKB Q96GD4 2/20 0.50
DDR1 Q08345 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL282308 0.87 CSF1R (0.70) CSF1RRAF1KDRPDGFRBKIT
SCHEMBL282549 0.78 CSF1R (0.72) CSF1RRAF1KDRPDGFRBKIT
SCHEMBL281954 0.76 CSF1R (0.70) CSF1RRAF1KDRPDGFRBKIT
SCHEMBL282705 0.76 KDR (0.61) CSF1RRAF1KDRPDGFRBKIT
SCHEMBL281915 0.74 CDK8 (0.48) RAF1KDRPDGFRBKITPDGFRA
SCHEMBL10073787 0.74 CSF1R (1.00) CSF1RRAF1KDRPDGFRBKIT
SCHEMBL22548172 0.74 CSF1R (0.83) CSF1RAURKB
SCHEMBL717412 0.73 CSF1R (0.77) CSF1RKDRPDGFRAFLT3AURKB
SCHEMBL22548456 0.72 CSF1R (1.00) CSF1RKDRPDGFRBKITPDGFRA
SCHEMBL22548194 0.70 CSF1R (0.82) CSF1RKDRAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2428506-A1 HETEROCYCLIC SUBSTITUTED ACARDITE DERIVATES AND USE THEREOF Jiangsu Provincial Institute Of Materia Medica Co. (CN) 2012-03-14 EP claimed