SCHEMBL28195201

SCHEMBL28195201

N#CC(C(=O)c1ccccc1)C(O)(C(=O)O)C(O)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.40
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ALKBH5 Q6P6C2 1/20 0.35
TSHR P16473 4/20 0.34
MDM2 Q00987 1/20 0.34
ALPG P10696 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PGR P06401 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
HTR2A P28223 1/20 0.32
HRH1 P35367 1/20 0.32
KCNH2 Q12809 1/20 0.32
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
DAO P14920 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27782158 0.73 LMNA (0.47) LMNACES2CES1TDP1L3MBTL1
SCHEMBL12373167 0.73 TDP1 (0.44) LMNACES2CES1TDP1L3MBTL1
SCHEMBL740027 0.73 CES1 (0.45) LMNACES2CES1TDP1L3MBTL1
SCHEMBL7342834 0.70 LMNA (0.52) LMNACES2CES1TDP1L3MBTL1
SCHEMBL28262205 0.69 LMNA (0.47) LMNACES2CES1TDP1L3MBTL1
Water SCHEMBL468373 0.69 CES1 (0.60) LMNACES2CES1TDP1L3MBTL1
SCHEMBL10741256 0.69 TDP1 (0.47) LMNACES2CES1TDP1L3MBTL1
Water SCHEMBL10705607 0.68 CES1 (0.44) LMNACES2CES1TDP1L3MBTL1
SCHEMBL23091851 0.68 TDP1 (0.50) LMNACES2CES1TDP1L3MBTL1
SCHEMBL408412 0.68 TDP1 (0.50) LMNACES2CES1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311892-A Preparation method of chiral pyrrolopyrimidine compound 正大天晴药业集团股份有限公司 2019-02-05 CN disclosed
CN-108699063-A Synthesis process of luccotinib 正大天晴药业集团股份有限公司 2018-10-23 CN disclosed
CN-107513069-A The preparation method of chiral Pyrrolopyrimidine compounds 正大天晴药业集团股份有限公司 2017-12-26 CN disclosed