SCHEMBL28196403

SCHEMBL28196403

COc1cccc(-c2[c]cccc2CN(C)C)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 6/20 0.41
SLC6A2 P23975 5/20 0.41
SLC6A3 Q01959 4/20 0.41
GRM5 P41594 1/20 0.41
HSD17B2 P37059 2/20 0.39
DYRK1A Q13627 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
HTR2A P28223 1/20 0.38
BACE1 P56817 1/20 0.38
MAOB P27338 1/20 0.38
CYP2D6 P10635 1/20 0.37
CALM1 P0DP23 1/20 0.37
CAMKK2 Q96RR4 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9070549 0.78 CLK4 (0.41) HSD17B2DYRK1ACLK4MAOBCYP2D6
SCHEMBL6048529 0.77 BACE1 (0.58) SLC6A4SLC6A2SLC6A3GRM5CLK4
SCHEMBL7843209 0.76 DYRK1A (0.45) DYRK1ACLK4MAOBCYP2D6ALDH1A1
SCHEMBL3411791 0.76 CYP1A1 (0.45) DYRK1ACLK4MAOBCYP2D6
SCHEMBL5506754 0.76 DYRK1A (0.45) DYRK1ACLK4MAOBCYP2D6
Hydrochloric Acid SCHEMBL6048554 0.75 BACE1 (0.57) SLC6A4SLC6A2SLC6A3GRM5CLK4
SCHEMBL9430884 0.75 DYRK1A (0.44) DYRK1ACLK4MAOBCYP2D6
SCHEMBL2377417 0.75 HDAC4 (0.55) DYRK1ACLK4CYP2D6
SCHEMBL4090309 0.71 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3HTR2AALDH1A1
SCHEMBL12472636 0.69 NPC1 (0.51) MAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017037-B 6 substituted aryl amino methyl tetrahydro naphthaline derivatives or its esters, and its production and use 复旦大学 2018-01-19 CN disclosed