SCHEMBL2819642

SCHEMBL2819642

COCCCCN1C(=O)[C@@H](C)Oc2cc(C(F)(F)F)c(C(=O)O)cc21

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
REN P00797 3/20 0.41
PPARG P37231 6/20 0.39
CYP3A4 P08684 2/20 0.37
CYP2C19 P33261 2/20 0.37
ALDH1A1 P00352 3/20 0.35
THRB P10828 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP2C9 P11712 1/20 0.34
LIPC P11150 1/20 0.33
LIPG Q9Y5X9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2239578 0.91 REN (0.41) RENPPARGCYP3A4CYP2C19ALDH1A1
SCHEMBL2242992 0.85 REN (0.43) RENPPARGCYP3A4CYP2C19ALDH1A1
SCHEMBL2820607 0.85 REN (0.47) RENPPARGCYP3A4CYP2C19ALDH1A1
SCHEMBL2243744 0.84 CYP3A4 (0.44) RENPPARGCYP3A4CYP2C19ALDH1A1
SCHEMBL2820593 0.82 REN (0.41) RENPPARGCYP3A4CYP2C19ALDH1A1
SCHEMBL12354040 0.82 POLB (0.36) RENPPARGCYP3A4CYP2C19ALDH1A1
SCHEMBL12352905 0.82 POLB (0.36) RENPPARGCYP3A4CYP2C19ALDH1A1
SCHEMBL2241986 0.81 REN (0.41) RENPPARGCYP3A4CYP2C19ALDH1A1
SCHEMBL2239580 0.80 REN (0.41) RENCYP2C19ALDH1A1MEN1KMT2A
SCHEMBL2245159 0.79 REN (0.34) RENPPARGCYP3A4CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8389511-B2 Bicyclic heterocyclic derivative DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2013-03-05 US disclosed
EP-2243779-A1 BICYCLIC HETEROCYCLIC DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2010-10-27 EP disclosed