SCHEMBL28197895

SCHEMBL28197895

FC(F)(F)c1cc(Br)n(-c2ccccc2)n1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.63
PTGS2 P35354 5/20 0.47
PDPK1 O15530 1/20 0.45
CYP1A2 P05177 2/20 0.44
KCNJ6 P48051 1/20 0.44
KCNJ5 P48544 1/20 0.44
KCNJ3 P48549 1/20 0.44
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NR3C2 P08235 1/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KLKB1 P03952 1/20 0.42
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323665 0.83 PTGS2 (0.53) PTGS1PTGS2PDPK1CYP2C9
SCHEMBL4830325 0.82 GRN (0.59) ALDH1A1SMN1; SMN2
SCHEMBL537395 0.80 PTGS1 (0.65) PTGS1PTGS2PDPK1CYP1A2KCNJ6
SCHEMBL7570850 0.80 PTGS1 (0.65) PTGS1PTGS2PDPK1CYP1A2ALDH1A1
SCHEMBL31625278 0.79 PDPK1 (0.53) PTGS1PTGS2PDPK1
SCHEMBL15478687 0.79 PTGS1 (0.63) PTGS1PTGS2PDPK1CYP1A2KCNJ6
SCHEMBL4978131 0.79 PTGS1 (0.63) PTGS1PTGS2PDPK1CYP1A2KCNJ6
SCHEMBL4666357 0.79 PTGS1 (0.63) PTGS1PTGS2PDPK1CYP1A2KCNJ6
SCHEMBL28157524 0.79 PTGS1 (0.68) PTGS1PTGS2PDPK1CYP1A2KCNJ6
SCHEMBL1012734 0.79 PTGS1 (0.63) PTGS1PTGS2PDPK1CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107567452-A Imidazopyrazine and pyrazolopyrimidine and their purposes as ampa receptor conditioning agent 詹森药业有限公司 2018-01-09 CN disclosed