SCHEMBL28198225

SCHEMBL28198225

O=C1c2cccc3c(N4CCOCC4)ccc(c23)C(=O)N1CCCO

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.71
HDAC3 O15379 3/20 0.71
HDAC1 Q13547 3/20 0.71
HDAC8 Q9BY41 2/20 0.71
HDAC11 Q96DB2 2/20 0.71
NCOR2 Q9Y618 2/20 0.71
HDAC2 Q92769 2/20 0.71
MEN1 O00255 12/20 0.69
KMT2A Q03164 12/20 0.69
MAPT P10636 4/20 0.69
RAB9A P51151 4/20 0.69
NPC1 O15118 2/20 0.69
AVPR1A P37288 1/20 0.69
HDAC10 Q969S8 1/20 0.63
L3MBTL1 Q9Y468 6/20 0.62
MAPK1 P28482 5/20 0.62
CRHBP P24387 4/20 0.62
CRHR2 Q13324 4/20 0.62
HTT P42858 3/20 0.62
POLB P06746 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22699960 0.93 MEN1 (0.80) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL28198224 0.89 MEN1 (0.86) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL28474023 0.86 MEN1 (0.69) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL12696859 0.86 HDAC3 (0.80) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL19327047 0.86 MEN1 (0.80) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL28197565 0.86 HDAC6 (0.64) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL12660423 0.85 HDAC3 (0.70) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL28203805 0.85 HDAC6 (0.70) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL12660402 0.84 HDAC6 (0.66) HDAC6HDAC3HDAC1HDAC8HDAC11
SCHEMBL12660336 0.84 HDAC6 (0.66) HDAC6HDAC3HDAC1HDAC8HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107698571-B Naphthalimide-coumarin DNA targeting double-intercalator, synthesis and application thereof 大连理工大学 2020-07-14 CN disclosed
CN-107698571-A Naphthalimide-coumarin DNA targeting double-intercalator, synthesis and application thereof 大连理工大学 2018-02-16 CN disclosed