SCHEMBL28199169

SCHEMBL28199169

CCC(=O)OC1CC=C[C@@H]1C(=O)OC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.33
CHRM2 P08172 2/20 0.33
CHRM4 P08173 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28199159 0.77 NFKB1 (0.40) NFKB1NFKB2RELA
SCHEMBL28039500 0.77 NFKB1 (0.40) NFKB1NFKB2RELA
SCHEMBL9836729 0.73 CHRM2 (0.38) CHRM2CHRM4CHRM1CHRM3
SCHEMBL7224503 0.68
SCHEMBL31472759 0.68 MAPK1 (0.36) MAPK1
SCHEMBL2535414 0.67 MAPK1 (0.42) MAPK1CHRM2CHRM1CHRM3NFKB1
SCHEMBL8603668 0.66 CHRM2 (0.37) CHRM2CHRM4CHRM1CHRM3
SCHEMBL28199171 0.66 MAPK1 (0.34) MAPK1
SCHEMBL13947268 0.64 NFKB1 (0.37) MAPK1NFKB1NFKB2RELA
SCHEMBL11227713 0.64 MAPT (0.37) MAPK1CHRM2CHRM1CHRM3NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143212-B Tripeptide epoxy ketone protease inhibitors 欧尼斯治疗公司 2018-02-23 CN disclosed