SCHEMBL28201225

SCHEMBL28201225

Cc1ccc(C#N)c(F)c1N

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
EGLN2 Q96KS0 4/20 0.38
POLB P06746 1/20 0.37
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
TRPV4 Q9HBA0 1/20 0.35
AR P10275 4/20 0.34
NOTUM Q6P988 1/20 0.34
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
MBOAT4 Q96T53 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17651309 0.83 TRPV4 (0.42) TSHREGLN2ALDH1A1KDM4EUSP2
SCHEMBL16382688 0.80 TSHR (0.44) TSHRPOLBALDH1A1KDM4EUSP2
SCHEMBL410450 0.80 TSHR (0.44) TSHREGLN2ALDH1A1TRPV4AR
SCHEMBL13199476 0.78 TSHR (0.43) TSHREGLN2POLBALDH1A1KDM4E
SCHEMBL11562734 0.78 POLB (0.50) TSHRPOLBALDH1A1KDM4EUSP2
SCHEMBL22684010 0.78 TRPV4 (0.38) EGLN2ALDH1A1KDM4EUSP2TRPV4
SCHEMBL30629031 0.78 POLB (0.50) TSHRPOLBALDH1A1KDM4EUSP2
SCHEMBL30432017 0.78 TRPV4 (0.38) EGLN2ALDH1A1KDM4EUSP2TRPV4
SCHEMBL17545789 0.77 TSHR (0.41) TSHREGLN2ALDH1A1KDM4ETRPV4
SCHEMBL1222533 0.75 TSHR (0.40) TSHREGLN2ALDH1A1TRPV4AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105339355-B Novel CYP17 inhibitor/antiandrogen 奥赖恩公司 2018-02-27 CN disclosed