SCHEMBL28201286

SCHEMBL28201286

[CH2]c1c(NC(=O)OC(C)(C)C)cnn1CCBr

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
CNR2 P34972 1/20 0.34
IDO1 P14902 2/20 0.33
BRD9 Q9H8M2 1/20 0.33
CYP17A1 P05093 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
MAPK14 Q16539 1/20 0.33
BRD4 O60885 1/20 0.32
METAP1 P53582 1/20 0.32
NAMPT P43490 1/20 0.32
GPR139 Q6DWJ6 1/20 0.32
SCD O00767 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
ABL1 P00519 1/20 0.32
SRC P12931 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18209904 0.82 CNR2 (0.37) GSK3BDYRK1ACNR2IDO1BRD9
SCHEMBL2173526 0.74 MAPK1 (0.41) GSK3BDYRK1ACNR2IDO1BRD9
SCHEMBL24255779 0.73 GSK3B (0.37) GSK3BDYRK1ACNR2IDO1BRD9
SCHEMBL18283999 0.72 CYP17A1 (0.39) GSK3BDYRK1ACNR2IDO1BRD9
SCHEMBL22322779 0.72 CNR2 (0.40) GSK3BDYRK1ACNR2BRD9CYP17A1
SCHEMBL22952416 0.72 GSK3B (0.39) GSK3BDYRK1ACNR2IDO1BRD9
SCHEMBL23009294 0.72 ATR (0.40) GSK3BDYRK1AIDO1BRD9HDAC3
SCHEMBL18366036 0.72 GSK3B (0.39) GSK3BDYRK1ACNR2IDO1BRD9
SCHEMBL25833918 0.71 CNR2 (0.38) GSK3BDYRK1ACNR2IDO1BRD9
SCHEMBL21164202 0.70 GSK3B (0.37) GSK3BDYRK1ACNR2IDO1BRD9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107646036-A Pyrazole derivatives useful as inhibitors of 5-lipoxygenase activating protein (F L AP) 阿斯利康(瑞典)有限公司 2018-01-30 CN disclosed