SCHEMBL28201498

SCHEMBL28201498

Fc1ccccc1Nc1nccc(-c2ccc3cn[nH]c3c2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 6/20 0.56
CLK4 Q9HAZ1 6/20 0.56
CDK2 P24941 5/20 0.56
CLK1 P49759 4/20 0.56
CLK2 P49760 5/20 0.53
DYRK1B Q9Y463 3/20 0.53
CDK1 P06493 2/20 0.51
RET P07949 2/20 0.51
CCNB2 O95067 1/20 0.51
CCNB1 P14635 1/20 0.51
CCNB3 Q8WWL7 1/20 0.51
CDK4 P11802 1/20 0.50
SYK P43405 4/20 0.46
SMO Q99835 1/20 0.46
CLK3 P49761 2/20 0.46
FGFR1 P11362 4/20 0.46
MAPK1 P28482 2/20 0.45
DAPK3 O43293 2/20 0.45
PRKD3 O94806 2/20 0.45
MAP4K4 O95819 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28856408 0.84 DYRK1A (0.64) DYRK1ACLK4CDK2CLK1CLK2
SCHEMBL28201500 0.81 CLK4 (0.58) DYRK1ACLK4CDK2CLK1CLK2
SCHEMBL28200962 0.80 DYRK1A (0.53) DYRK1ACLK4CDK2CLK1CLK2
SCHEMBL27114006 0.78 CCNB2 (0.52) CDK2CDK1RETCCNB2CCNB1
SCHEMBL29481867 0.78 DYRK1A (0.62) DYRK1ACLK4CDK2CLK1CLK2
SCHEMBL28727089 0.78 DYRK1A (0.62) DYRK1ACLK4CDK2CLK1CLK2
SCHEMBL14519531 0.77 CDK4 (0.57) CDK2CDK1RETCCNB2CCNB1
SCHEMBL27116075 0.77 CCNB2 (0.55) CDK2CDK1RETCCNB2CCNB1
SCHEMBL28201525 0.76 ABL1 (0.63) DYRK1ACLK4CDK2CLK1CLK2
SCHEMBL3760002 0.76 SYK (0.60) DYRK1ACLK4CDK2CLK1CLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107721991-B A kind of 6- (pyrimidine-4-yl) -1H- indazole derivative and its preparation method and application 南方医科大学中西医结合医院 2019-10-18 CN disclosed
CN-107721991-A A kind of 6 (base of pyrimidine 4) 1H indazole derivatives and its preparation method and application 南方医科大学中西医结合医院 2018-02-23 CN disclosed