SCHEMBL28201525

SCHEMBL28201525

Clc1cccc(Nc2nccc(-c3ccc4cn[nH]c4c3)n2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.63
BCR P11274 1/20 0.63
PRKCA P17252 1/20 0.63
PRKCD Q05655 1/20 0.63
CAMK2D Q13557 6/20 0.61
CDK2 P24941 5/20 0.58
CLK1 P49759 2/20 0.58
DYRK1A Q13627 2/20 0.58
CLK4 Q9HAZ1 2/20 0.58
CLK2 P49760 1/20 0.57
DYRK1B Q9Y463 1/20 0.57
PLK1 P53350 1/20 0.57
SYK P43405 1/20 0.55
BTK Q06187 1/20 0.55
CSNK2A1 P68400 2/20 0.54
CDK4 P11802 2/20 0.53
CDK1 P06493 2/20 0.53
SMG1 Q96Q15 2/20 0.53
MAPT P10636 2/20 0.53
NPC1 O15118 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28201500 0.87 CLK4 (0.58) ABL1BCRPRKCAPRKCDCAMK2D
SCHEMBL27115512 0.84 CLK1 (0.61) CDK2CLK1DYRK1ACLK4CLK2
SCHEMBL28856408 0.83 DYRK1A (0.64) ABL1PRKCDCAMK2DCDK2CLK1
SCHEMBL27115203 0.81 ABL1 (0.61) ABL1BCRPRKCAPRKCDCAMK2D
SCHEMBL3246795 0.81 NUDT1 (0.62) ABL1BCRPRKCAPRKCDCAMK2D
SCHEMBL3760002 0.80 SYK (0.60) ABL1PRKCAPRKCDCAMK2DCDK2
SCHEMBL3510842 0.79 ABL1 (0.75) ABL1BCRPRKCAPRKCDCAMK2D
SCHEMBL27114009 0.79 CAMK2D (0.63) ABL1BCRPRKCAPRKCDCAMK2D
SCHEMBL3513778 0.78 CAMK2D (0.73) ABL1BCRPRKCAPRKCDCAMK2D
SCHEMBL30847308 0.78 SMO (0.60) CAMK2DCDK2CLK1DYRK1ACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107721991-B A kind of 6- (pyrimidine-4-yl) -1H- indazole derivative and its preparation method and application 南方医科大学中西医结合医院 2019-10-18 CN disclosed
CN-107721991-A A kind of 6 (base of pyrimidine 4) 1H indazole derivatives and its preparation method and application 南方医科大学中西医结合医院 2018-02-23 CN disclosed