SCHEMBL28201638

SCHEMBL28201638

C[Si](C)(C)Cn1ccnn1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.42
FOLH1 Q04609 1/20 0.33
DPP4 P27487 1/20 0.33
CYP1A1 P04798 1/20 0.31
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL251196 0.74
SCHEMBL10424811 0.73 CYP19A1 (0.48) CYP19A1FOLH1DPP4CYP1A1
SCHEMBL11361006 0.73 CYP19A1 (0.48) CYP19A1FOLH1DPP4CYP1A1
SCHEMBL2384020 0.72 CYP19A1 (0.36) CYP19A1
SCHEMBL33258 0.70
SCHEMBL13088477 0.70
SCHEMBL11898438 0.69 CYP19A1 (0.44) CYP19A1FOLH1CYP1A1
SCHEMBL10374 0.69 CYP19A1 (0.34) CYP19A1
SCHEMBL5333181 0.69
SCHEMBL6483599 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108558871-A Novel tricyclic compound as anticancer agent 百时美施贵宝公司 2018-09-21 CN disclosed
CN-106029663-B Tricyclic compounds as anticancer agents 百时美施贵宝公司 2018-06-01 CN disclosed
CN-107709322-A Tricyclic compound as anticancer 百时美施贵宝公司 2018-02-16 CN disclosed