SCHEMBL10374

SCHEMBL10374

C[Si](C)(C)CCOCn1ccnn1

nearest known ligand 0.34

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2659461 0.80 CYP19A1 (0.33) CYP19A1
SCHEMBL7265318 0.79 CYP19A1 (0.38) CYP19A1
SCHEMBL6250570 0.76
SCHEMBL11617 0.74 FDPS (0.33)
SCHEMBL29092717 0.74 MEN1 (0.43)
Ammonia Solution, Strong SCHEMBL27898568 0.73 FDPS (0.32)
SCHEMBL3303673 0.71
SCHEMBL15032983 0.70 DGAT1 (0.32)
SCHEMBL28201638 0.69 CYP19A1 (0.42) CYP19A1
SCHEMBL4606038 0.68 DGAT1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 92 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12357615-B2 Compositions for the treatment of brain tumors KEMBI THERAPEUTICS PTY LTD (AU) 2025-07-15 US disclosed
US-20220370415-A1 COMPOSITIONS FOR THE TREATMENT OF BRAIN TUMORS KEMBI THERAPEUTICS PTY LTD (AU) 2022-11-24 US disclosed
WO-2019182743-A1 COMPOSITIONS FOR THE TREATMENT OF BRAIN TUMORS INNOCRIN PHARMACEUTICALS, INC. (US) 2019-09-26 WO disclosed
EP-3483147-A1 METALLOENZYME INHIBITOR COMPOUNDS Innocrin Pharmaceuticals, Inc. (US) 2019-05-15 EP disclosed
EP-3483147-A1 METALLOENZYME INHIBITOR COMPOUNDS Innocrin Pharmaceuticals, Inc. (US) 2019-05-15 EP disclosed
CN-108707177-A 20- triazol radical -20- hydroxyls-pregnant steroid derivatives and preparation method thereof and medical usage 中国药科大学 2018-10-26 CN disclosed
EP-2638021-B1 1-(6,7-Bis(difluoromethoxy)naphthalen-2-yl)-2-methyl-1-(1H-1,2,3-triazol-4-yl)propan-1-ol as inhibitor of CYP17 for the treatment of androgen dependent diseases like prostate cancer INNOCRIN PHARMACEUTICALS INC (US) 2018-09-26 EP disclosed
US-20180221364-A1 METALLOENZYME INHIBITOR COMPOUNDS INNOCRIN PHARMACEUTICALS, INC. 2018-08-09 US disclosed
US-20180221364-A1 METALLOENZYME INHIBITOR COMPOUNDS INNOCRIN PHARMACEUTICALS, INC. 2018-08-09 US disclosed
US-20180221364-A1 METALLOENZYME INHIBITOR COMPOUNDS INNOCRIN PHARMACEUTICALS, INC. 2018-08-09 US disclosed
US-6255305-B1 PSYCHOLOGICAL DISORDERS MERCK SHARP & DOHME LIMITED (GB) 2001-07-03 US disclosed
US-6200975-B1 FOR COGNITION ENHANCEMENT THERAPY MERCK SHARP & DOHME LIMITED (GB) 2001-03-13 US disclosed
EP-1070066-A1 SUBSTITUTED 1,2,4-TRIAZOLO 3,4-a]PYRIDAZINE MERCK SHARP & DOHME LTD. (GB) 2001-01-24 EP disclosed
WO-2000027849-A2 THERAPEUTIC POLYMORPHS OF A GABA-A ALPHA-5 INVERSE AGONIST AND PAMOATE FORMULATIONS OF THE SAME MERCK & CO., INC. (US) 2000-05-18 WO disclosed
WO-2000027382-A2 COMBINATION OF A GABA-A ALPHA 5 INVERSE AGONIST AND COX-2 INHIBITOR, NSAID, ESTROGEN OR VITAMIN E MERCK & CO., INC. (US) 2000-05-18 WO disclosed
EP-0986562-A1 SUBSTITUTED 1,2,4-TRIAZOLO 3,4-A]PHTHALAZINE DERIVATIVES AS GABA ALPHA 5 LIGANDS MERCK SHARP & DOHME LTD. (GB) 2000-03-22 EP disclosed
WO-1999043677-A1 SUBSTITUTED 1,2,4-TRIAZOLO[3,4-a]PYRIDAZINE MERCK SHARP & DOHME LIMITED (GB) 1999-09-02 WO disclosed
EP-0915875-A2 SUBSTITUTED TRIAZOLO-PYRIDAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 1999-05-19 EP disclosed
WO-1998050385-A1 SUBSTITUTED 1,2,4-TRIAZOLO[3,4-a]PHTHALAZINE DERIVATIVES AS GABA ALPHA 5 LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1998-11-12 WO disclosed
WO-1998004559-A2 SUBSTITUTED TRIAZOLO-PYRIDAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1998-02-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180221364-A1 METALLOENZYME INHIBITOR COMPOUNDS MMEL1, GPX1, MPO CYP19A1 898/4885
US-20220370415-A1 COMPOSITIONS FOR THE TREATMENT OF BRAIN TUMORS NR3C2, NR3C1, CRH CYP19A1 1262/4885
US-12357615-B2 Compositions for the treatment of brain tumors NR3C2, NR3C1, CRH CYP19A1 1262/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.