SCHEMBL28201899

SCHEMBL28201899

Cc1c(C(=O)O)cc(-c2cccc(N)c2)cc1C(=O)O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.66
MAOA P21397 1/20 0.52
KMT2A Q03164 5/20 0.49
KDM4E B2RXH2 4/20 0.49
MEN1 O00255 4/20 0.49
TDP1 Q9NUW8 3/20 0.49
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48
GFER P55789 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
MAP4K4 O95819 2/20 0.47
PLK4 O00444 1/20 0.47
EGFR P00533 1/20 0.47
ROS1 P08922 1/20 0.47
PIM1 P11309 1/20 0.47
AXL P30530 1/20 0.47
FLT3 P36888 1/20 0.47
FRK P42685 1/20 0.47
MAP4K2 Q12851 1/20 0.47
NTRK3 Q16288 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26981146 0.82 MCL1 (0.75) MCL1MAOAKMT2AKDM4EMEN1
SCHEMBL27786187 0.81 PTPN1 (0.58) MCL1AKR1C2AKR1C1ACMSDALDH1A1
SCHEMBL28201890 0.80 TDP1 (0.53) MCL1KMT2AKDM4EMEN1TDP1
SCHEMBL27639373 0.80 MCL1 (0.57) MCL1MAOAKMT2AKDM4EMEN1
SCHEMBL2796864 0.79 MCL1 (0.53) MCL1MAOAMEN1MAP4K4PLK4
SCHEMBL28479099 0.79 MCL1 (1.00) MCL1MAOAKMT2AKDM4EMEN1
SCHEMBL28201920 0.79 AKR1C2 (0.48) MCL1KMT2AKDM4EMEN1AKR1C2
SCHEMBL27786189 0.77 ACMSD (0.53) MCL1KMT2AKDM4EMEN1TDP1
SCHEMBL27692105 0.77 POLB (0.51) MCL1KMT2AKDM4EMEN1TDP1
SCHEMBL27846422 0.77 KMT2A (0.59) MCL1KMT2AKDM4EMEN1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164113-B Pyrroloamide inhibitors 艾伯维公司 2018-03-02 CN claimed
CN-105164113-B Pyrroloamide inhibitors 艾伯维公司 2018-03-02 CN disclosed