SCHEMBL28205243

SCHEMBL28205243

FC(F)(F)c1ccccc1-c1ccncn1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 12/20 0.53
CYP3A4 P08684 11/20 0.53
KMO O15229 2/20 0.51
CYP2C19 P33261 12/20 0.49
CYP2D6 P10635 9/20 0.49
ALOX15 P16050 6/20 0.49
HSD17B10 Q99714 5/20 0.49
ALDH1A1 P00352 3/20 0.49
MAPK1 P28482 2/20 0.49
CLK4 Q9HAZ1 1/20 0.47
TSHR P16473 2/20 0.47
HIF1A Q16665 1/20 0.47
TDP1 Q9NUW8 2/20 0.47
KDM4E B2RXH2 1/20 0.44
USP2 O75604 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
P2RX7 Q99572 1/20 0.43
HSD11B1 P28845 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28273372 0.82 CYP3A4 (0.39) CYP1A2CYP3A4KMOCYP2C19CYP2D6
SCHEMBL10601314 0.80 MAPK9 (0.43) CYP2D6CLK4
SCHEMBL4166620 0.79 TGFBR1 (0.56) CYP1A2CYP3A4KMOCYP2C19CYP2D6
SCHEMBL31211635 0.79 TGFBR1 (0.56) CYP1A2CYP3A4KMOCYP2C19CYP2D6
SCHEMBL30090604 0.79 TGFBR1 (0.56) CYP1A2CYP3A4KMOCYP2C19CYP2D6
SCHEMBL28239064 0.77 MAPK10 (0.43) CYP1A2CYP3A4KMOCLK4P2RX7
SCHEMBL6220344 0.76 ACP1 (0.40) CYP1A2CYP3A4KMOCYP2C19CYP2D6
SCHEMBL28461573 0.76 CYP3A4 (0.53) CYP1A2CYP3A4KMOCYP2C19CYP2D6
SCHEMBL30141958 0.76 NPC1 (0.46) KMT2A
SCHEMBL28296072 0.76 NPC1 (0.46) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107759571-A Inhibitors of influenza viruses replication and its application method and purposes 广东东阳光药业有限公司 2018-03-06 CN disclosed