SCHEMBL28206403

SCHEMBL28206403

C[C@@H](c1ccccc1)n1nccc1C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.49
ALDH1A1 P00352 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
FAAH O00519 1/20 0.42
ALOX5 P09917 1/20 0.40
KDM5A P29375 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
MAPK1 P28482 1/20 0.40
BRD2 P25440 1/20 0.39
BRD3 Q15059 1/20 0.39
BRDT Q58F21 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28348292 0.89 ALDH1A1 (0.53) BRD4ALDH1A1TDP1FAAHKDM5A
SCHEMBL24966152 0.89 ALDH1A1 (0.53) BRD4ALDH1A1TDP1FAAHKDM5A
SCHEMBL23234281 0.87 BRD4 (0.46) BRD4ALDH1A1TDP1FAAHMAPK1
SCHEMBL24966148 0.87 BRD4 (0.46) BRD4ALDH1A1TDP1FAAHMAPK1
SCHEMBL24966182 0.86 BRD4 (0.45) BRD4ALDH1A1TDP1FAAHMAPK1
SCHEMBL24966867 0.83 BRD4 (0.46) BRD4ALDH1A1TDP1FAAHMAPK1
SCHEMBL24966866 0.83 BRD4 (0.43) BRD4ALDH1A1TDP1FAAHMAPK1
SCHEMBL24966063 0.82 BRD4 (0.42) BRD4ALDH1A1TDP1FAAHMAPK1
SCHEMBL2307447 0.81 NR3C2 (0.48) ALDH1A1
SCHEMBL24966075 0.81 BRD4 (0.41) BRD4ALDH1A1TDP1FAAHKDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107690281-A Cystic fibrosis transmembrane transduction modulator modulators 弗特克斯药品有限公司 2018-02-13 CN disclosed