Phenylacetylene

Phenylacetylene

SCHEMBL28207262

C#Cc1ccc2ccoc2c1.C#Cc1ccccc1

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.43
CYP2A6 P11509 2/20 0.40
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35
CYP2C9 P11712 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
NFKB1 P19838 1/20 0.35
MAOA P21397 1/20 0.35
ACHE P22303 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PTPN1 P18031 1/20 0.35
HTR1B P28222 3/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15441267 0.76 CYP2A6 (0.66) CYP2A6CYP1A1CYP1B1CYP2C9KDM4E
SCHEMBL506960 0.72 CYP2A6 (0.71) CYP2A6CYP2C9KDM4ECYP3A4CYP2D6
SCHEMBL96525 0.72 CYP2A6 (0.46) GRM5CYP2A6CYP2C9KDM4ECYP3A4
SCHEMBL891207 0.70 DYRK1A (0.48) CYP2A6CYP2C9KDM4ECYP3A4CYP2D6
SCHEMBL30646399 0.70 DYRK1A (0.48) CYP2A6CYP2C9KDM4ECYP3A4CYP2D6
Phenylacetylene SCHEMBL4297769 0.69
Phenylacetylene SCHEMBL1331558 0.69
Phenylacetylene SCHEMBL1331398 0.69
Phenylacetylene SCHEMBL4884 0.69
Phenylacetylene SCHEMBL1331408 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104945389-B A kind of mountain ketone colour contamination ketone compounds and its preparation method and application 中国科学院上海药物研究所 2018-04-13 CN disclosed