SCHEMBL28208196

SCHEMBL28208196

O=C(O)c1ccc(CN(CC2CC2)C(=O)c2ccc(Br)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.64
HDAC6 Q9UBN7 2/20 0.64
LPAR1 Q92633 16/20 0.61
LPAR5 Q9H1C0 16/20 0.61
PKM P14618 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16507443 0.84 HDAC1 (0.59) HDAC1HDAC6LPAR1LPAR5PKM
SCHEMBL16506463 0.76 LPAR1 (1.00) LPAR1LPAR5
SCHEMBL14720201 0.75 HDAC1 (0.52) HDAC1HDAC6LPAR1LPAR5PKM
SCHEMBL16506625 0.75 LPAR1 (1.00) LPAR1LPAR5
SCHEMBL16506976 0.75 LPAR1 (1.00) LPAR1LPAR5
SCHEMBL16506833 0.75 LPAR1 (1.00) LPAR1LPAR5
SCHEMBL16506837 0.75 LPAR1 (1.00) LPAR1LPAR5
SCHEMBL16507344 0.74 LPAR1 (1.00) LPAR1LPAR5
SCHEMBL16506601 0.74 LPAR1 (1.00) LPAR1LPAR5
SCHEMBL16506872 0.71 LPAR1 (1.00) LPAR1LPAR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105473548-B Amide derivatives as lpa receptor antagonist 武田药品工业株式会社 2018-03-23 CN disclosed