SCHEMBL28210973

SCHEMBL28210973

Cc1ccnnc1-c1cccnc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 11/20 0.62
CYP3A4 P08684 5/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 1/20 0.50
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP2E1 P05181 3/20 0.46
CYP2C9 P11712 3/20 0.46
CYP2B6 P20813 3/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
NPY5R Q15761 1/20 0.45
MAP2K4 P45985 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL221221 0.80 PDK1 (0.42) CYP2A6ALDH1A1KDM4EMAPTHPGD
SCHEMBL30385626 0.78 CYP2A6 (0.50) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL3613457 0.77 CYP2A6 (1.00) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL16826037 0.74 CYP2A6 (0.53) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL30385344 0.74 CYP2A6 (0.49) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL28277835 0.71 ADORA2A (0.46) CYP3A4KDM4E
SCHEMBL12258295 0.71 CYP2A6 (0.59) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL13910994 0.71 CYP2A6 (0.70) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL9137297 0.70 CYP2A6 (0.58) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL18104257 0.70 CYP2A6 (0.68) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105992767-B WNT pathway modulators 新加坡科技研究局 2019-06-21 CN disclosed
CN-106061974-B Maleimide derivatives as the conditioning agent of WNT approach 新加坡科技研究局 2018-04-20 CN disclosed