SCHEMBL28215433

SCHEMBL28215433

COc1cccc(C#CF)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.56
CA1 P00915 3/20 0.56
CA2 P00918 3/20 0.56
CA9 Q16790 3/20 0.56
CA12 O43570 2/20 0.56
CHRM2 P08172 1/20 0.50
CHRM1 P11229 1/20 0.50
CHRM3 P20309 1/20 0.50
FFAR1 O14842 1/20 0.49
ACHE P22303 1/20 0.48
CA7 P43166 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
HAO1 Q9UJM8 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6132140 0.89 GRM5 (0.66) GRM5CA1CA2CA9CA12
SCHEMBL30707880 0.89 GRM5 (0.66) GRM5CA1CA2CA9CA12
SCHEMBL25490057 0.86 GRM5 (0.54) GRM5CA1CA2CA9CA12
SCHEMBL29994376 0.83 GRM5 (0.56) GRM5CA1CA2CA9CA12
SCHEMBL7601866 0.83 GRM5 (0.56) GRM5CA1CA2CA9CA12
SCHEMBL4267103 0.83 CA12 (0.63) GRM5CA1CA2CA9CA12
SCHEMBL28397792 0.82 CA1 (0.58) GRM5CA1CA2CA9CA12
SCHEMBL8207581 0.82 GRM5 (0.54) GRM5CA1CA2CA9CA12
SCHEMBL27916593 0.82 GRM5 (0.54) GRM5CA1CA2CA9CA12
SCHEMBL24434459 0.82 GRM5 (0.54) GRM5CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107963996-B Method for preparing 3-trifluoromethyl isoxazole compound by one-pot method 江西师范大学 2021-06-11 CN disclosed
CN-108069918-B Method for preparing 3-difluoromethyl isoxazole compound by one-pot method 江西师范大学 2021-05-28 CN disclosed
CN-108069918-A Method for preparing 3-difluoromethyl isoxazole compound by one-pot method 江西师范大学 2018-05-25 CN disclosed
CN-107963996-A Method for preparing 3-trifluoromethyl isoxazole compound by one-pot method 江西师范大学 2018-04-27 CN disclosed