SCHEMBL28215935

SCHEMBL28215935

CCCCCn1cc(-c2ccnc(N)n2)c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.52
CNR2 P34972 5/20 0.49
GSK3B P49841 1/20 0.48
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
TLR8 Q9NR97 4/20 0.47
MKNK1 Q9BUB5 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
ICMT O60725 1/20 0.46
CNR1 P21554 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28215934 0.82 DYRK1A (0.55) DYRK1AGSK3BMKNK1MKNK2
SCHEMBL28507558 0.81 DYRK1A (0.75) DYRK1ACNR2GSK3BCA12CA1
SCHEMBL29870510 0.79 CDC7 (0.60) DYRK1AGSK3BMKNK1MKNK2
SCHEMBL5750318 0.79 CDC7 (0.60) DYRK1AGSK3BMKNK1MKNK2
Hydrochloric Acid SCHEMBL5749287 0.78 CDC7 (0.59) DYRK1AGSK3BMKNK1MKNK2
SCHEMBL19532488 0.77 MKNK2 (0.54) DYRK1ACNR2GSK3BCA12CA1
SCHEMBL15625751 0.74 CA12 (0.53) CNR2GSK3BCA12CA1CA2
SCHEMBL22585743 0.72 EGFR (0.49) GSK3BMKNK1MKNK2
SCHEMBL31278246 0.72 EGFR (0.49) GSK3BMKNK1MKNK2
SCHEMBL17542604 0.71 MKNK2 (0.53) DYRK1AGSK3BCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108218838-B Pyrimidine radicals indole derivatives and preparation method thereof and application in preparation of anti-tumor drugs 青岛海洋生物医药研究院股份有限公司 2019-07-23 CN disclosed
CN-108218838-A Pyrimidine radicals indole derivatives and preparation method thereof and application in preparation of anti-tumor drugs 青岛海洋生物医药研究院股份有限公司 2018-06-29 CN disclosed