SCHEMBL28217080

SCHEMBL28217080

Nc1ccc(C(=O)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.77

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 7/20 0.77
P2RX1 P51575 5/20 0.71
HDAC3 O15379 1/20 0.61
HDAC8 Q9BY41 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
MEN1 O00255 1/20 0.61
LMNA P02545 1/20 0.61
POLB P06746 1/20 0.61
PKM P14618 1/20 0.61
APEX1 P27695 1/20 0.61
KMT2A Q03164 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
JUN P05412 1/20 0.56
NFKB1 P19838 1/20 0.56
NFKB2 Q00653 1/20 0.56
RELA Q04206 1/20 0.56
TRPA1 O75762 1/20 0.56
MAPT P10636 1/20 0.55
TRPV1 Q8NER1 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL683803 0.91 PTGS1 (0.68) PTGS1P2RX1HDAC3HDAC8HDAC6
SCHEMBL678064 0.87 PTGS1 (0.77) PTGS1P2RX1HDAC3HDAC8HDAC6
SCHEMBL678654 0.87 PTGS1 (1.00) PTGS1HDAC3HDAC8HDAC6MEN1
SCHEMBL11307930 0.86 PTGS1 (0.76) PTGS1P2RX1MEN1LMNAKMT2A
SCHEMBL28329635 0.85 P2RX1 (0.64) PTGS1P2RX1HDAC3HDAC8HDAC6
SCHEMBL19638212 0.84 P2RX1 (0.71) PTGS1P2RX1HDAC3HDAC8HDAC6
SCHEMBL11799771 0.84 P2RX1 (0.71) P2RX1HDAC3HDAC8HDAC6MEN1
SCHEMBL23447713 0.83 P2RX1 (1.00) P2RX1HDAC3HDAC8HDAC6LMNA
SCHEMBL2914683 0.83 P2RX1 (0.74) P2RX1HDAC3HDAC8HDAC6LMNA
SCHEMBL7588013 0.82 PTGS1 (0.60) PTGS1P2RX1HDAC3HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108084096-A 2- phenyl pyrimidine classes compound, preparation method and medical usage 中国药科大学 2018-05-29 CN disclosed