SCHEMBL28217237

SCHEMBL28217237

CC(C)c1cccc([C@H](C)C2CC2)c1-n1ccnc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.43
ALOX15 P16050 2/20 0.43
CYP3A4 P08684 3/20 0.37
CYP11B2 P19099 3/20 0.35
USP1 O94782 1/20 0.35
WDR48 Q8TAF3 1/20 0.35
CYP11B1 P15538 2/20 0.35
IDO1 P14902 2/20 0.35
CYP1A2 P05177 1/20 0.35
GAA P10253 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP2A6 P11509 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28217238 1.00 TSHR (0.43) TSHRALOX15CYP3A4CYP11B2USP1
SCHEMBL928068 0.88 TSHR (0.48) TSHRALOX15CYP3A4CYP11B2USP1
Hydrochloric Acid SCHEMBL1819866 0.86 TSHR (0.47) TSHRALOX15CYP3A4CYP11B2USP1
Hydrochloric Acid SCHEMBL28362336 0.85 TSHR (0.46) TSHRALOX15CYP3A4CYP11B2USP1
Fluoride SCHEMBL28981521 0.85 TSHR (0.46) TSHRALOX15CYP3A4CYP11B2USP1
SCHEMBL28021700 0.83 TSHR (0.44) TSHRALOX15CYP3A4CYP11B2USP1
Pyridine SCHEMBL27763194 0.82 CYP3A4 (0.44) TSHRALOX15CYP3A4CYP11B2USP1
SCHEMBL28217261 0.82 DPP4 (0.36) TSHRALOX15CYP3A4CYP1A2HTR2C
SCHEMBL28217262 0.82 DPP4 (0.36) TSHRALOX15CYP3A4CYP1A2HTR2C
Boric Acid SCHEMBL28901108 0.81 TSHR (0.43) TSHRALOX15CYP3A4CYP11B2USP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108017559-B Benzene ring derivative and application thereof in medicine 四川海思科制药有限公司 2020-08-04 CN disclosed
CN-108017559-A Phenyl ring derivative and its application in medicine 四川海思科制药有限公司 2018-05-11 CN disclosed