SCHEMBL28217261

SCHEMBL28217261

CC(C)c1cccc([C@H](C)C2CC2)c1-n1cccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
GABRA1 P14867 3/20 0.35
TSHR P16473 3/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRB2 P47870 2/20 0.35
FAAH O00519 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.35
GABRB1 P18505 1/20 0.35
PTGS1 P23219 1/20 0.35
SLC6A2 P23975 1/20 0.35
HTR2C P28335 1/20 0.35
GABRA5 P31644 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28217262 1.00 DPP4 (0.36) DPP4NR1H2NR1H3GABRA1TSHR
SCHEMBL28217672 0.96 DPP4 (0.32) DPP4NR1H2NR1H3ANPEP
SCHEMBL28217673 0.96 DPP4 (0.32) DPP4NR1H2NR1H3ANPEP
SCHEMBL28045533 0.85 GABRA1 (0.46) DPP4NR1H2NR1H3GABRA1TSHR
SCHEMBL28217237 0.82 TSHR (0.43) TSHRCYP1A2CYP3A4HTR2CHTR2B
SCHEMBL28217238 0.82 TSHR (0.43) TSHRCYP1A2CYP3A4HTR2CHTR2B
SCHEMBL28217235 0.78 MEN1 (0.36) DPP4NR1H2NR1H3GABRA1TSHR
SCHEMBL28217232 0.78 MEN1 (0.36) DPP4NR1H2NR1H3GABRA1TSHR
SCHEMBL21154977 0.74 GABRA1 (0.40) DPP4NR1H2NR1H3GABRA1TSHR
SCHEMBL28217215 0.74 KCNQ2 (0.32) HTR2CHTR2BHIF1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108017559-B Benzene ring derivative and application thereof in medicine 四川海思科制药有限公司 2020-08-04 CN disclosed
CN-108017559-A Phenyl ring derivative and its application in medicine 四川海思科制药有限公司 2018-05-11 CN disclosed