SCHEMBL28217265

SCHEMBL28217265

NS(=O)(=O)c1ccc(-c2ccc(C(=O)N3CCN(c4ccccc4)CC3)cc2)cc1

nearest known ligand 0.92

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 12/20 0.92
CA2 P00918 12/20 0.92
CA9 Q16790 12/20 0.92
CA7 P43166 11/20 0.92
CA12 O43570 11/20 0.92
CA14 Q9ULX7 9/20 0.92
MEN1 O00255 3/20 0.74
KMT2A Q03164 3/20 0.74
SLC6A7 Q99884 2/20 0.74
POLB P06746 2/20 0.74
TP53 P04637 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28014906 0.89 CA1 (0.73) CA1CA2CA9CA7CA12
SCHEMBL8161635 0.86 SLC6A7 (1.00) CA1CA2CA9CA7CA12
SCHEMBL28217169 0.84 CA12 (0.69) CA1CA2CA9CA7CA12
SCHEMBL10721777 0.83 MEN1 (0.87) CA1CA2CA9CA7CA12
SCHEMBL14493373 0.83 CA12 (0.87) CA1CA2CA9CA7CA12
SCHEMBL5632669 0.80 SLC6A7 (0.67) CA1CA2CA9CA7CA12
SCHEMBL8595777 0.80 POLB (0.87) CA1CA2CA9CA7CA12
SCHEMBL3276407 0.79 MEN1 (0.74) CA1CA2CA9CA7CA12
SCHEMBL1711050 0.79 MEN1 (0.74) CA1CA2CA9CA7CA12
SCHEMBL3573771 0.77 SLC6A7 (0.81) MEN1KMT2ASLC6A7POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104817498-B Therapeutic compound and composition 安吉奥斯医药品有限公司 2018-06-01 CN disclosed
CN-104817498-A Therapeutic compounds and compositions AGIOS PHARMACEUTICALS INC 2015-08-05 CN disclosed
CN-102481300-B Therapeutic compounds and compositions AGIOS PHARMACEUTICALS INC 2015-04-15 CN disclosed