SCHEMBL282174

SCHEMBL282174

COc1cc2c(Oc3ccc(N)cc3)ccnc2cc1F

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 6/20 0.59
PDGFRB P09619 1/20 0.59
FGFR2 P21802 5/20 0.56
KDR P35968 5/20 0.54
MET P08581 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL167396 0.89 PDGFRA (0.74) PDGFRAPDGFRBFGFR2KDR
SCHEMBL901281 0.88 PDGFRA (0.68) PDGFRAPDGFRBFGFR2KDRMET
Hydrochloric Acid SCHEMBL23528156 0.88 PDGFRA (0.72) PDGFRAPDGFRBFGFR2KDR
SCHEMBL22188238 0.86 PDGFRA (0.55) PDGFRAPDGFRBFGFR2KDRMET
Fluorobenzene SCHEMBL28724473 0.85 FGFR2 (0.65) PDGFRAPDGFRBFGFR2KDRMET
SCHEMBL4141203 0.84 FGFR2 (0.60) PDGFRAPDGFRBFGFR2KDR
SCHEMBL14540576 0.84 PDGFRA (0.62) PDGFRAPDGFRBFGFR2KDR
SCHEMBL13980801 0.83 PDGFRA (0.60) PDGFRAPDGFRBFGFR2KDR
SCHEMBL21201045 0.82 PDGFRA (0.59) PDGFRAPDGFRBFGFR2KDR
SCHEMBL166914 0.82 AXL (0.67) PDGFRAPDGFRBFGFR2KDRMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8957087-B2 Heterocyclic substituted acardite derivate and application thereof Jiangsu Provincial Institute of Materia Medica Co., Ltd. (CN) 2015-02-17 US disclosed
EP-2428506-B1 HETEROCYCLIC SUBSTITUTED ACARDITE DERIVATES AND USE THEREOF NANJING LUYESIKE PHARMACEUTICAL CO LTD (CN) 2014-03-05 EP disclosed
EP-2428506-A1 HETEROCYCLIC SUBSTITUTED ACARDITE DERIVATES AND USE THEREOF Jiangsu Provincial Institute Of Materia Medica Co. (CN) 2012-03-14 EP disclosed
US-20120053192-A1 Heterocyclic Substituted Acardite Derivate and Application Thereof NANJING LUYESIKE PHARMACEUTICAL CO., LTD. (CN) 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053192-A1 Heterocyclic Substituted Acardite Derivate and Application Thereof H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, IDH1, CA7 PDGFRA 1115/4885PDGFRB 1549/4885FGFR2 367/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.