SCHEMBL28217671

SCHEMBL28217671

CC(C)c1cc(C=O)cc(C(C)C2CC2)c1N

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TYR P14679 1/20 0.32
EGFR P00533 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2B6 P20813 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28217668 1.00 TYR (0.32) TYREGFRCYP1A2CYP3A4CYP2B6
SCHEMBL6284758 0.84 TYR (0.41) TYREGFRCYP1A2CYP3A4CYP2B6
SCHEMBL19704411 0.81 CYP1A2 (0.46) EGFRCYP1A2CYP3A4CYP2B6
SCHEMBL28258800 0.81 CYP1A2 (0.46) EGFRCYP1A2CYP3A4CYP2B6
SCHEMBL19704222 0.78 CYP1A2 (0.39) TYREGFRCYP1A2CYP3A4CYP2B6
SCHEMBL28258767 0.78 CYP1A2 (0.39) TYREGFRCYP1A2CYP3A4CYP2B6
SCHEMBL28217729 0.76 FABP3 (0.35)
SCHEMBL28217282 0.76 FABP3 (0.35)
SCHEMBL21543066 0.74 SRC (0.37) TYREGFRCYP1A2CYP3A4CYP2B6
SCHEMBL17972912 0.70 GABRA1 (0.39) CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108017559-B Benzene ring derivative and application thereof in medicine 四川海思科制药有限公司 2020-08-04 CN disclosed
CN-108017559-A Phenyl ring derivative and its application in medicine 四川海思科制药有限公司 2018-05-11 CN disclosed