SCHEMBL28219641

SCHEMBL28219641

CN(C)C1CCN(c2ncnc(Cl)n2)C1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.47
DYRK1A Q13627 1/20 0.46
HRH4 Q9H3N8 4/20 0.45
HRH3 Q9Y5N1 2/20 0.43
JAK2 O60674 3/20 0.42
JAK3 P52333 3/20 0.42
PTPN11 Q06124 1/20 0.41
HDAC6 Q9UBN7 1/20 0.37
EGLN2 Q96KS0 1/20 0.37
PDE10A Q9Y233 2/20 0.37
BRAF P15056 1/20 0.37
CHRM1 P11229 1/20 0.37
HRH1 P35367 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28543291 0.82 MAP4K4 (0.53) MAP4K4DYRK1AHRH4HRH3JAK2
SCHEMBL28220125 0.80 MAP4K4 (0.46) MAP4K4DYRK1AHRH4HRH3JAK2
SCHEMBL14812129 0.78 MAP4K4 (0.37) MAP4K4JAK2JAK3PTPN11
SCHEMBL19251255 0.77 DYRK1A (0.47) MAP4K4DYRK1AHRH4HRH3JAK2
SCHEMBL20507807 0.77 SUV39H2 (0.43) MAP4K4DYRK1AHRH4HRH3PTPN11
SCHEMBL1775585 0.73 HRH4 (0.58) MAP4K4HRH4HRH3JAK2JAK3
SCHEMBL13806026 0.73 DYRK1A (0.55) MAP4K4DYRK1AHRH4HRH3
SCHEMBL13806029 0.73 DYRK1A (0.55) MAP4K4DYRK1AHRH4HRH3
SCHEMBL1774527 0.73 HRH4 (0.58) MAP4K4HRH4HRH3JAK2JAK3
SCHEMBL12487715 0.72 DYRK1A (0.54) MAP4K4DYRK1AHRH4HRH3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108135175-A Bicyclic compounds and their use for inhibition of SUV39H2 肿瘤疗法科学股份有限公司 2018-06-08 CN disclosed