Bromide

Bromide

SCHEMBL28224569

Br.C=CCc1cccc(OC)c1

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 3/20 0.50
CHRM3 known ✓ P20309 3/20 0.50
SIGMAR1 known ✓ Q99720 1/20 0.47
ALDH1A1 P00352 3/20 0.58
CYP3A4 P08684 2/20 0.58
TP53 P04637 1/20 0.58
ALOX15 P16050 1/20 0.58
TSHR P16473 1/20 0.58
ALOX12 P18054 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
TAAR1 Q96RJ0 3/20 0.53
IDO1 P14902 2/20 0.53
AGXT P21549 2/20 0.53
PPARG P37231 1/20 0.53
PPARD Q03181 1/20 0.53
PPARA Q07869 1/20 0.53
CHRM1 P11229 3/20 0.50
CMA1 P23946 1/20 0.49
ALOX5 P09917 1/20 0.49
AR P10275 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29382328 0.98 ALDH1A1 (0.60) ALDH1A1CYP3A4TP53ALOX15TSHR
SCHEMBL2091147 0.98 ALDH1A1 (0.60) ALDH1A1CYP3A4TP53ALOX15TSHR
Water SCHEMBL28328781 0.87 ALDH1A1 (0.49) ALDH1A1CYP3A4TP53ALOX15TSHR
Phenol SCHEMBL28310738 0.87 MAOB (0.51) ALDH1A1CYP3A4TP53ALOX15TSHR
SCHEMBL29212064 0.83 ALDH1A1 (0.45) ALDH1A1CYP3A4TP53ALOX15TSHR
SCHEMBL28567450 0.82 ALDH1A1 (0.60) ALDH1A1CYP3A4TP53ALOX15TSHR
SCHEMBL8305017 0.82 TAAR1 (0.58) TAAR1IDO1AGXTCHRM2CHRM1
SCHEMBL8406148 0.82 ALDH1A1 (0.44) ALDH1A1CYP3A4TP53ALOX15TSHR
SCHEMBL3503547 0.81 TAAR1 (0.56) TAAR1IDO1AGXTCHRM2CHRM1
SCHEMBL248658 0.81 CHRM2 (0.57) ALDH1A1SMN1; SMN2TAAR1IDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108101826-A Indoles substituted alkylamine class compound and application thereof 华东理工大学 2018-06-01 CN disclosed