SCHEMBL28228697

SCHEMBL28228697

CN1CCN(c2ccc(Nc3ncc(C(=O)O)cn3)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LCK P06239 4/20 0.60
MAPK14 Q16539 4/20 0.60
KDR P35968 2/20 0.59
ALK Q9UM73 2/20 0.57
BRD4 O60885 4/20 0.56
EGFR P00533 1/20 0.55
SYK P43405 2/20 0.54
CDK4 P11802 3/20 0.54
CCND1 P24385 3/20 0.54
CCND2 P30279 1/20 0.54
CCND3 P30281 1/20 0.54
STAT6 P42226 1/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
CHEK1 O14757 1/20 0.53
INSR P06213 1/20 0.53
MAP4K1 Q92918 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4492001 0.88 SYK (0.62) LCKMAPK14KDRALKBRD4
SCHEMBL28228708 0.84 SYK (0.54) SYKCDK4CCND1CCND2CCND3
SCHEMBL4721744 0.83 LCK (0.81) LCKMAPK14KDRBRD4NPC1
SCHEMBL31163120 0.83 BRD4 (0.75) BRD4EGFR
SCHEMBL19496537 0.81 LCK (0.59) LCKMAPK14KDRALKBRD4
SCHEMBL29037749 0.81 ALK (0.69) LCKMAPK14ALKBRD4EGFR
SCHEMBL29037828 0.81 EGFR (0.60) ALKBRD4EGFRSYKCDK4
SCHEMBL2961783 0.81 EGFR (0.60) LCKMAPK14KDRALKEGFR
SCHEMBL2951233 0.81 ALK (0.62) LCKMAPK14ALKBRD4EGFR
SCHEMBL30463630 0.81 ALK (0.65) LCKMAPK14KDRALKBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108299312-A One group of pyridine derivatives and its application in preparation of anti-tumor drugs 郑州大学第附属医院 2018-07-20 CN disclosed