SCHEMBL28228708

SCHEMBL28228708

O=C(O)c1cnc(Nc2ccc(N3CCNCC3)cc2)nc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.54
STAT6 P42226 1/20 0.53
MAPK8 P45983 1/20 0.53
MAPK9 P45984 1/20 0.53
MAPK10 P53779 1/20 0.53
CDK4 P11802 9/20 0.52
CCND1 P24385 5/20 0.52
CCND3 P30281 4/20 0.52
CCND2 P30279 2/20 0.52
CDK2 P24941 5/20 0.51
CCNA2 P20248 4/20 0.51
CCNE1 P24864 2/20 0.50
CDK1 P06493 1/20 0.50
CCNB1 P14635 1/20 0.50
CDK6 Q00534 3/20 0.49
FGFR1 P11362 2/20 0.49
FGFR2 P21802 2/20 0.49
FGFR4 P22455 2/20 0.49
FGFR3 P22607 2/20 0.49
CCNE2 O96020 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4488495 0.88 SYK (0.62) SYKSTAT6MAPK8MAPK9MAPK10
SCHEMBL28228697 0.84 LCK (0.60) SYKSTAT6CDK4CCND1CCND3
SCHEMBL21275499 0.79 PLK4 (0.57) MAPK8MAPK9CDK4CCND1CDK2
SCHEMBL30459671 0.77 CDK4 (0.53) STAT6CDK4CCND1CCND3CCND2
SCHEMBL598515 0.76 ALDH1A1 (0.72) ALDH1A1USP2TSHRHSD17B10
SCHEMBL28227975 0.75 SYK (0.48) SYKSTAT6MAPK8MAPK9MAPK10
Hydrochloric Acid SCHEMBL4652111 0.75 ALDH1A1 (0.70) ALDH1A1USP2TSHRHSD17B10
SCHEMBL7064739 0.74 SYK (0.60) SYKSTAT6MAPK8MAPK9MAPK10
SCHEMBL3590138 0.74 PDGFRB (0.62) SYKSTAT6CDK4CCND1CCND3
SCHEMBL598464 0.74 POLB (0.65) ALDH1A1USP2TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108299312-A One group of pyridine derivatives and its application in preparation of anti-tumor drugs 郑州大学第附属医院 2018-07-20 CN disclosed